एम.व्ही.पी. समाजाचे

के. टी. एच. एम. महाविद्यालय

(के.आर.टी. कला, बी.एच. वाणिज्य, ए.एम. विज्ञान महाविद्यालय.)

MVP SAMAJ'S

K.T.H.M. COLLEGE, Nashik

(K.R.T. Arts, B.H. Commerce and A.M. Science College.)

Faculty Profile

 
Faculty Name :
Dr. Raghunath Baban Toche
Specialization :
Organic chemistry
Date Of Birth :
01/06/1959
Email :
Phone :
0253 2518373
Mobile :
9420692839
Address :
blessings, Professor Colony, Hanumanwadi Panchawati, Nashik-422003

  Qualification :

Sr. No Degree University / Institution Grade Year of Passing Specialization
1 B.Sc. University of Pune O 1979 Chemistry 
2 M.Sc. University of Pune B+ 1981 Org. Chemistry 
3 Ph.D. University of Pune -- 2001 Org.Chemistry 
4 DHE University of Pune B+ 1985 Education 

 

 Experience :

Name  & Address of Employer Post Held Period of service Nature of Duties
Garware Polyester Pvt Ltd, Ambad  R & D Chemist 1981-82 R & D 
KTHM College, Nashik-02 Jr. College Teacher 1982-84 Teaching 
ASC College, Deolali Camp Lecturer  1984- 95 Teaching 
KTHM College, Nashik-02 Lecturer   1996-2005 Tecahing & Research 
KTHM College, Nashik-02 Associate Professor  2006-17 Tecahing & Research 

 

 Papers In International Refereed Journals :

Sr. No.

Title of Research paper

1

A Facile Synthesis of 5-benzoylcytosine derivatives, Organic Preparations &Procedures International; 30(3), 1998, 367-372. R.B.Toche, M.N.Jachak, T.S. Dalvi

Organic Preparations &Procedures International 30 (3), 367 1998

2

A Facile Synthesis of 5-Benzoylcytosine Derivatives RB Toche, MN Jachak, TS Dalvi, RW Sabnis, H Junek, T Kappe Organic preparations and procedures international 30 (3), 367-372 1998

3

Novel Synthesis of Fused Pyrano Quinolone, Coumarins and Pyridones; J. Heterocycl. chem. 36, 467, 1999 ISSN: 1943-5193 R.B.Toche, M.N.Jachak Journal of Heterocyclic Chemistry 36, 467, 1999

4

Synthesis of novel pyrano fused quinolones, coumarins, and pyridones RB Toche, MN Jachak, RW Sabnis, T Kappe 1999 Journal of heterocyclic chemistry 36 (2), 467-471

5

Phase Transfer catalyst in Grindstone synthesis of 3-oxopropanitrile in water: One pot synthesis of polysubstituted amino thiophene derivatives; R.B.Toche, S.B. Kanwade, M.P. Shinde Indian Journalof heterocyclic Chemistry 21, 33,  2001

6

A convenient route for the synthesis of 4-aryl & 4-aminopyrimidines,  MN Jachak, CD Tantak, RB Toche, Monatshefte für Chemie 135, 1529, 2004

7

A convenient route for the synthesis of 4-aryl-and 4-aminopyrimidines MN Jachak, CD Tantak, RB Toche, NS Badgujar Monatshefte für Chemie/Chemical Monthly 135 (12), 1529-1538 2004

8

Friedländer condensation of 5-aminopyrazole-4-carbaldehydes with reactive α-methylene ketones: Synthesis of pyrazolo [3, 4-b] pyridines MN Jachak, AB Avhale, CD Tantak, RB Toche, C Reidlinger, Journal of heterocyclic chemistry 42 (7), 1311-1319 2005

9

Formation of oxiranes during the preparation of aroylacetonitriles RB Toche, MN Jachak, NS Badgujar, AB Avhale, DB Kendre Organic preparations and procedures international 37 (4), 405-408 2005

10

Formation of Oxiranes during the Preparation of Aroylacetonitriles

R.B.Toche, M.N. Jachak, N. S.Badgujar, D.K. Kendre Organic Preparations Procedures International 37 (4), 405  2005

11

Synthesis and evaluation of insect repellent activity of 4-amino-5-(4-bromobenzoyl)-3-ethyl-2 (1H)-pyrimidone, on Setophilus oryzae (Coleo curculeonidae)

R Toche, V Medhane, A Desai, A Avhale, D Kendre, M Jachak Journal of the Indian Chemical Society 83 (10), 1039-1040   2006

12

Synthesis of novel benzochromene, benzoquinoline, benzochromenopyrimidine and pyrimidobenzoquinoline derivatives MN Jachak, DB Kendre, AB Avhale, RB Toche, VJ Medhane

Organic preparations and procedures international 38 (3), 313-324 2006

13

A convenient route for the synthesis of pyrazolo [3, 4-d] pyrimidine, pyrazolo [3, 4-b][1, 6] naphthyridine and pyrazolo [3, 4-b] quinoline derivatives MN Jachak, AB Avhale, VJ Medhane, RB Toche Journal of heterocyclic chemistry 43 (5), 1169-1175

14

ORGN 96-Design, synthesis and study of novel blue light-emitting benzo [h] quinolines as organic antennas for luminescence resonance energy transfer

MN Jachak, DB Kendre, RB Toche, RW Sabnis ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 232; 2006

15

Synthesis and evaluation of insect repellent activity of 4-amino-5-(4-bromo benzoyl)-3-ethyl -2-(1H)- pyrimidone onsetophilusoryzae (Coleo curculeonidae)

Journal of Indian Chemical Society 43, 1306, RB Toche, M. Kazi 2006

16

Synthesis of novel Dipyrazolo [3, 4-b: 3, 4-d] pyridines and study of their fluorescence behavior DB Kendre, RB Toche, MN Jachak Tetrahedron 63 (45), 11000-11004

17

Synthesis of pyrazolo-annelated heterocyclic ring compounds such as pyrazolo [3, 4-b] pyridines and pyrazolo [4′, 3′: 5, 6]-pyrido [2, 3-d] pyrimidines MN Jachak, AB Avhale, RB Toche, RW Sabnis Journal of Heterocyclic Chemistry 44 (2), 343-347 2007

18

Synthesis of fused pyrimidines from amines and cyclic β-formylesters

RB Toche, BK Ghotekar, MA Kazi, DB Kendre, MN Jachak Tetrahedron 63 (34), 8157-8163 2007

19

A novel synthesis of benzo [h] quinolines and study of their fluorescence properties

MN Jachak, DB Kendre, AB Avhale, RB Toche, RW Sabnis Journal of Heterocyclic Chemistry 44 (6), 1525-1528 2007

20

Facile synthesis of novel fused pyrimidines RB Toche, BK Ghotekar, MA Kazi, DB Kendre, MN Jachak, RW Sabnis ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 233 2007

21

Synthesis of pyrazolo [3, 4-b] pyridines using ammonium acetate as green reagent in multi-component reactions MN Jachak, AB Avhale, BK Ghotekar, DB Kendre, RB Toche

Journal of Heterocyclic Chemistry 45 (4), 1221-1224 2008

22

Synthesis of pyrazolo [3, 4-b] pyridines and attachment of amino acids and carbohydrate as linkers DB Kendre, RB Toche, MN Jachak Journal of Heterocyclic Chemistry 45 (5), 1281-1286 2008

23

Effect of substituents on absorption and fluorescence properties of pyrazolo [3, 4-b] pyrrolo [2, 3-d] pyridines

BK Ghotekar, MA Kazi, MN Jachak, RB Toche Canadian Journal of Chemistry 86 (11), 1070-1076 2008

24

Michael addition of dimedone with α, β-unsaturated ketones: Synthesis of quinoline and chromene derivatives DB Kendre, RB Toche, MN Jachak Journal of Heterocyclic Chemistry 45 (3), 667-671 2008

25

An efficient synthesis of pyrazolo [3, 4-b] pyrrolo [2, 3-d] pyridines from 5-aminopyrazoles and cyclic β-keto ester RB Toche, BK Ghotekar, DB Kendre, MA Kazi, MN Jachak Journal of Heterocyclic Chemistry 45 (6), 1711-1717 2008

26

Synthesis of 4-cyano-and 5-aminopyrazoles and deamination of 5-aminopyrazoles

RB Toche, MA Kazi, MN Jachak Organic Preparations and Procedures International 40 (6), 551-556 2008

27

New Approach for the Synthesis of Pyrido [1, 2-a] pyrimidines

RB Toche, BK Ghotekar, MA Kazi, SP Patil, MN Jachak Scholarly Research Exchange 2008

28

New Approach for the Synthesis of Pyrido [1, 2-a] pyrimidines

RB Toche, BK Ghotekar, MA Kazi, SP Patil, MN Jachak Scholarly Research Exchange 2008

29

New one-step synthesis of pyrazolo [1, 5-a] pyrimidine and pyrazolo [1, 5-a] quinazoline derivatives via multicomponent reactions BK Ghotekar, MN Jachak, RB Toche

Journal of Heterocyclic Chemistry 46 (4), 708-713 2009

30

Synthesis and study of the fluorescent behavior of 3-pyridinecarbonitriles MN Jachak, SM Bagul, BK Ghotekar, RB Toche Monatshefte für Chemie-Chemical Monthly 140 (6), 655 2009

31

Fluorescence properties of donor acceptor chromophores on newly synthesized pyridine-3-carbonitriles RB Toche, MA Kazi, BK Ghotekar, SM Bagul, CD Tantak, MN Jachak

Journal of fluorescence 19 (6), 1119 2009

32

Vilsmeier–Haack formylation of acetonitrile revisited: Synthesis of novel pyrazolo [1, 5-a] pyrimidines and triazolo [1, 5-a] pyrimidine MG Ghagare, DR Birari, DP Shelar, RB Toche, MN Jachak Journal of Heterocyclic Chemistry 46 (2), 327-331  2009

33

Synthesis of cytosine derivatives and study of their alkylation under mild conditions

DR Birari, MG Ghagare, MA Kazi, SM Bagul, BK Ghotekar, RB Toche, Organic Preparations and Procedures International 41 (6), 515-532 2009

34

Synthesis of benzohetero [3, 2-a] pyrimidines using cyclic β-keto lactone as a building block RB Toche, BK Ghotekar, MA Kazi, MN Jachak Monatshefte für Chemie-Chemical Monthly 140 (2), 235 2009

35

Synthesis of new quinoline fused heterocycles such as benzo [h]-1, 6-naphthyridines and pyrazolo [4, 3-c] quinolines BK Ghotekar, MG Ghagare, RB Toche, MN Jachak

Monatshefte für Chemie-Chemical Monthly 141 (2), 169-175 2010

36

Synthesis of pyrazolopyridine 3-carboxylates by Friedlander condensation

RB Toche, DC Bhavsar, MA Kazi, SM Bagul, MN Jachak Journal of Heterocyclic Chemistry 47 (2), 287-291 2010

37

Synthesis of novel spiro-oxazino-quinoline derivatives and study of their photophysical properties BS Rane, MA Kazi, SM Bagul, DP Shelar, RB Toche, MN Jachak

Journal of fluorescence 20 (1), 415-420 2010

38

Synthesis of novel benzo [h][1, 6] naphthyridine derivatives from 4-aminoquinoline and cyclic β-ketoester RB Toche, BP Pagar, RR Zoman, GB Shinde, MN Jachak

Tetrahedron 66 (27), 5204-5211 2010

39

Synthesis and molluscicidal activities of quinolone substituted pyrazoline and isoxazoline derivatives. RB Toche, MA Kazi, MN Jachak, AE Desai Journal of Applied Sciences Research, 637-641 2010

40

Synthesis and fluorescence properties of donor-acceptor-substituted novel dipyrazolo [3, 4-b: 3′, 4′-d] pyridines (DPP) MN Jachak, SM Bagul, DR Birari, MG Ghagare, MA Kazi, RB Toche, Journal of fluorescence 20 (3), 787-796 2010

41

New chromogenic spray reagent for detection and identification of carbosulfan

K Kulkarni, D Shinde, D Mane, R Toche, M Garad JPC-Journal of Planar Chromatography-Modern TLC 23 (5), 373-375 2010

42

Synthesis of quinolone substituted pyrazoles, isoxazoles and pyridines as a potential blue luminophors RB Toche, MA Kazi, SP Patil, SB Kanawade, MN Jachak

Journal of fluorescence 20 (5), 1129-1137 2010

43

Synthesis of uracil derivatives and their alkylation: an approach to peptide non-nucleic acid monomers MN Jachak, DR Birari, RB Toche, MG Ghagare, SM Bagul Monatshefte für Chemie-Chemical Monthly 141 (4), 451-459 2010

44

Novel and Efficient Synthesis of Pyrimidine Derivatives MG Ghagare, DR Birari, DP Shelar, RB Toche, MN Jachak Synthetic Communications® 40 (11), 1580-1587 2010

45

A novel synthetic approach towards pyrazole-4-carboxamides using N-(3-(dimethylamino)-2-formylacryloyl) formamide RB Toche, MN Jachak, MG Ghagare, DR Birari, RV Rote, MA Kazi, SM Jachak, Monatshefte für Chemie-Chemical Monthly 141 (5), 569-576 2010

46

Industrial Application of the Forster Reaction: Novel One-Pot Synthesis of Cinacalcet Hydrochloride, a Calcimimetic Agent; GB Shinde, NC Niphade, SP Deshmukh, RB Toche, VT Mathad, Organic Process Research & Development 15 (2), 455-461   2011

47

Novel synthesis of 2-aminoquinoline-3-carbaldehyde, benzo [b][1, 8] naphthyridines and study of their fluorescence behavior DP Shelar, DR Birari, RV Rote, SR Patil, RB Toche, MN Jachak Journal of Physical Organic Chemistry 24 (3), 203-211    2011

48

Arylbenzo [h][1, 6] naphthyridine derivatives: synthesis and photophysical properties; RB Toche, RA Janrao, SM Bagul, SP Patil, BP Pagar, PS Nikam Journal of fluorescence 21 (4), 1617-1624    2011

49

Synthesis and fluorescence investigation of differently substituted benzo [b][1, 8] naphthyridines: Interaction with different solvents and bovine serum albumin (BSA); DP Shelar, SR Patil, RV Rote, RB Toche, MN Jachak Journal of fluorescence 21 (3), 1033-1047  2011

50

Aminothiophenedicarboxamides and dicyanothiopheneacetamides as effective synthetic molluscicides against Indoplanorbis exustus snail

SB Kanawade, RB Toche, SP Patil, AE Desai, SS Bhamare; European journal of medicinal chemistry 46 (9), 4682-4686  2011

51

Synthesis of benzo [3, 4-h][1, 6] naphthyridines via Friedländer condensation with active methylenes; RV Rote, SM Bagul, DP Shelar, SR Patil, RB Toche, MN Jachak

Journal of Heterocyclic Chemistry 48 (2), 301-307; 2011

52

Novel synthetic protocol toward pyrazolo [3, 4-h]-[1, 6] naphthyridines via Friedlander condensation of new 4-aminopyrazolo [3, 4-b] pyridine- 5-carbaldehyde with reactive α-methylene ketones MN Jachak, SM Bagul, MA Kazi, RB Toche Journal of Heterocyclic Chemistry 48 (2), 295-300 2011

53

Effect of donor-acceptor chromophores on photophysical properties of newly synthesized Pyrazolo-pyrrolo-pyrimidines (PPP) RV Rote, DP Shelar, SR Patil, SS Shinde, RB Toche, MN Jachak Journal of fluorescence 21 (1), 453-459 2011

54

Synthesis of nicotinonitrile derivatives and study of their photophysical properties

RB Toche, MA Kazi, PS Nikam, DC Bhavsar Monatshefte für Chemie-Chemical Monthly 142 (3), 261-269

2011

55

Use of sodium salt of cyclic β-formylester for synthesis of dihydro-2H-furo [2, 3-d] pyrazolo [3, 4-b] pyridines and pyrazolo [3, 4-b] pyrrolo [2, 3-d] pyridines

SP Patil, RB Toche Monatshefte für Chemie-Chemical Monthly 142 (11), 1193-1201

56

Effect of Specific Solute-Solvent Interaction and Electron Donor-Acceptor Substituents of Novel Pyrazolo Naphthyridines on Fluorescence SR Patil, DP Shelar, RV Rote, RB Toche, MN Jachak Journal of fluorescence 21 (1), 461-471 2011

57

Unusual finding of pyrethroid insecticide used for leopard hunting—a case report

K Kulkarni, D Shinde, D Mane, R Toche, M Garad JPC-Journal of Planar Chromatography-Modern TLC 24 (5), 445-446 2011

58

Synthetic utility of a heterocyclic o-aminoaldehyde: synthesis of  pyrazolo pyridopyrimidines, pyrazolonaphthyridines, and pyrazolopyrimidonaphthyridinones

SM Bagul, DR Birari, MG Ghagare, RB Toche, MN Jachak 2011

Monatshefte für Chemie-Chemical Monthly 142 (2), 169-175, 2011

59

Phase transfer catalyst in grindstone synthesis of 3-oxopropanenitrile: One pot synthesis of polysubstituted amino thiophenes SP Patil, SB Kanawade, MP Shinde, RB Toche

Indian Journal of Heterocyclic Chemistry 21 (1), 33-36 2011

60

New chromogenic spray reagent for detectionand identification of hydrogen cyanamide, KV Kulkarni, DB Shind, DV Mane, RB Toche, Global Journal Analytical Chemistry; 2(1), 2011, 46-49. 2011

61

Synthesis of new thieno [2, 3-d] pyrimidines, thieno [3, 2-e] pyridines, and thieno [2, 3-d][1, 3] oxazines,SB Kanawade, SP Patil, PS Nikam, SA Gangurde, MN Jachak, RB Toche. Journal of Heterocyclic Chemistry 49 (2), 363-369  2012

62

Expedient approach for the synthesis of novel indenothiophene derivatives

SP Patil, MA Kazi, SB Kanawade, PS Nikam, MN Jachak, RB Toche

Monatshefte für Chemie-Chemical Monthly 143 (2), 317-323   2012

63

Synthesis of Pyrazolopyridine Annulated Heterocycles and Study the Effect of Substituents on Photophysical Properties; SP Patil, DP Shelar, RB Toche

Journal of fluorescence 22 (1), 31-41     2012

64

Synthetic tactics of new class of 4-aminothieno [2, 3-d] pyrimidine-6-carbonitrile derivatives acting as antimicrobial agents SB Kanawade, RB Toche, DP Rajani

European journal of medicinal chemistry 64, 314-320   2013

65

Sulfamic Acid–Mediated, Efficient, One-Pot Synthesis of Novel 5-Substituted 1, 3, 4-Thiadiazol-2-ylcarbamoyl Aliphatic Amide Acid Derivatives and Facile Synthesis of Cyclic Amides; RB Toche, RA Janrao, SA Gangurde, PS Nikam; Synthetic Communications 43 (18), 2527-2535  2013

66

An Efficient Microwave-assisted Suzuki Cross-coupling Reactions on Quinoline Derivatives in Water and Study the Electronic Effects Thereof

R Toche, R Janrao International Journal of Scientific and Research Publications, Volume 3, Issue 8, August 2013 1 ISSN 2250-3153, 2013

67

Microwave-assisted synthesis of fused tricyclic pyrazino [1, 2-a] indole derivatives

R Toche, S Chavan, R Janrao Monatshefte für Chemie-Chemical Monthly 145 (9), 1507-1512 2014

68

Syntheses of New Unsymmetrical 2, 5-Disubstituted-1, 3, 4-oxadiazoles and 1, 2, 4-Triazolo [3, 4-b]-1, 3, 4-thiadiazoles Bearing Thieno [2, 3-c] pyrazolo Moiety

SP Patil, SB Kanawade, DC Bhavsar, PS Nikam, SA Gangurde, RB Toche

Journal of Heterocyclic Chemistry 51 (2), 368-373   2014

69

Syntheses of New Unsymmetrical 2, 5-Disubstituted-1, 3, 4-oxadiazoles and 1, 2, 4-Triazolo [3, 4-b]-1, 3, 4-thiadiazoles Bearing Thieno [2, 3-c] pyrazolo Moiety

SP Patil, SB Kanawade, DC Bhavsar, PS Nikam, SA Gangurde, RB Toche

Journal of Heterocyclic Chemistry 51 (2), 368-373  2014

70

Synthesis of Polysubstituted Pyrazolo [3, 4-b] pyridine-3-Carbohydrazide and Pyrazolo [3, 4-d] pyridazine Derivatives, DC Bhavsar, PS Nikam, SA Gangurde, RB Toche

Journal of Heterocyclic Chemistry 51 (3), 635-641   2014

71

Synthesis and Study the Effect of Donor-Acceptor Substituent on Fluorescence Behavior of Thieno [3, 2-c] pyridine Derivatives, RB Toche, SN Chavan, Journal of fluorescence 24 (2), 285-293    2014

72

New Synthesis and Reactions of Ethyl 5-amino-4-cyano -1-phenyl -1H- pyrazole -3-carboxylate; SA Gangurde, SB Kanawade, PS Nikam, DC Bhavsar, RB Toche

Journal of Heterocyclic Chemistry;  51 (4), 883-890   2014

73

A green approach for the synthesis of organic heterocyclic compounds such as pyrazolo [3, 4-b] pyridine derivatives, SA Chaudhari, VM Patil, MM Chavan, SV Patil, RB Toche, MN Jachak; International journal of pharmaceutical Research & Development (IJPRD), 6(10) 87-95; 2014

74

Microwave-assisted synthesis of fused tricyclic

pyrazino[1,2-a]indole derivatives Raghunath Toche,  Sunil Chavan , Ravindra Janrao  Monatsh Chem (2014) 145:1507–1512   2014

75

Synthesis, Characterization of β-amino ketone Complexes and Study of their Antibacterial Activity R Watpade, P Tandale, M Shinde, P Dhondge, R Toche, 2015

76

Rapid determination of alpha tocopherol in olive oil adulterated with sunflower oil by reversed phase high-performance liquid chromatography, SM Bakre, DK Gadmale, RB Toche, VB Gaikwad, Journal of food science and technology 52 (5), 3093-3098  2015

77

An efficient and safe process for the preparation of ticagrelor, a platelet aggregation inhibitor via resin-NO2 catalyzed formation of triazole ring

GB Shinde, PK Mahale, SA Padaki, NC Niphade, RB Toche, VT Mathad, SpringerPlus 4 (1), 493 2015

78

Synthesis, characterization and antimicrobial evaluation of novel urea, sulfonamide and acetamide 3, 4-dihydropyrazino [1, 2-a] indol-1 (2H)-one derivatives, RB Toche, RA Janrao, Arabian Journal of Chemistry   doi.org/10.1016/j.arabjc.2015.08.034  2015

79

Synthesis and evaluation of antimicrobial and antitubercular activity of arylidene hydrazines of indenothieno[2,3-d]pyrimidine, Chemistry & biology interface;

RB Toche, P Nikam, Chemistry & Biology 5 (4), 246-257  2015

80

The Use of Pinner Type Reaction for the Synthesis of New Indeno [2, 1-c] pyridine-4-carbonitrile Derivatives; PS Nikam, SP Patil, SB Kanawade, SA Gangurde, M Rathi, RB Toche Journal of Heterocyclic Chemistry 52 (1), 150-155   2015

81

Reactions of ketene dithioacetal for a new versatile synthesis of 4, 5-substituted 3-aminothiophene-2-carboxylate derivatives; SM Chavan, RB Toche, VM Patil, PB Aware, PS Patil, Journal of Sulfur Chemistry 37 (4), 426-437   2016

82

In vitro Antimicrobial Evaluation of 3-Aminothiophene-2-carboxylates

PARW Satish Chavan,Raghunath Toche*, Avinash Bhole, Vasant Patil

Journal of Chemical and Pharmaceutical Research, 8 (4), 198-201   2016

83

Sucrose and KF quenching system for solution phase parallel synthesis

S Chavan, R Watpade, R Toche,  SpringerPlus 5 (1), 1058    2016

84

Synthesis and Characterization of Novel Semicarbazone Derivatives of Disubstituted N-arylmaleimides, S Chaudhari, V Patil, S Chavan, K Dingore, S Patil,

R Toche, M Jachak, Der Pharma Chemica , 8(7) 66-73; 2016

85

Aminothiophene Carboxylates as Effective Molluscicidal Agents against Fresh Water Pond Snail Lymnaea stagnalis in Maharashtra, India

S Chavan, R Toche, A Desai, V Patil, P Aware, M Jachak Journal of Pharmaceutical, Chemical and Biological Sciences, ISSN: 2348-7658 , 2016

 

86

Synthesis and Characterization of Pd (II) Schiff Base Metal Complexes

,ISSN 0975-413X CODEN (USA): PCHHAX, MP Shinde, RB Toche, SM Chavan, PJ Tambade, Der Pharma Chemica, 2016, 8(10):287-293  2016

87

Simple route for the synthesis of pyrido [1, 2-a] pyrimidine derivatives , ISSN 0975-413X CODEN (USA): PCHHAX, Der Pharma Chemica, 2016, 8(3):146-151

RB Toche, PB Aware, SM Chavan, VM Patil, PS Patil, 2016

88

Determination of Ethanol Content in Medicated Syrups: A Comparison among Distillation, Titration and GC Methods

raghunath Toche, Shobha Borhade, Balasaheb Daundkar and Bhausaheb More Chemical Science Transactions ISSN:2278-3458 2016, 5(1), 248-252

89

In vitro Antimicrobial Evaluation of 3-Aminothiophene-2-carboxylates, Satish Chavan1,2, Raghunath Toche Journal of Chemical and Pharmaceutical Research, 2016, 8(4):198-201

90

Substituent Effect on Absorption and Fluorescence Properties of Thieno[3, 2-c]Pyridine Derivatives, Sunil N. Chavan1,3 & Raghunath B. Toche1,3 & Satish M. Chavan2,3,

Journal of Fluorescence,  DOI 10.1007/s10895-017-2026-1; 2017

 

 Papers In National Refereed Journals :

Sr. No Name of Author(s) Full Title of the Paper Journal Name Volume No Issue No. Year of Publication From Page To Page (pp)
               

 Papers In International Conference :

1

Synthesis and photo physical properties of 3-pyridine carbonitrile

 

International conference in Chemical Education

 

Homi Bhabha Centre for Science Education

Mumbai,

 

Nov.12-14, 2010

2

Synthesis of 3,5-disubstitutd cytosine derivatives;

36th Annual Conventional of Chemists ,

Indian Chemical Society

Calcutta

16-12-1999

3

Synthesis of cytosine derivatives

International Conference on Heterocyclic Chemistry

Rajasthan University

Jaipur

Dec.16-19, 2006

4

Arylation of Unprotected quinoline derivatives by  Suzuki Miyaura Reaction in Water

International Science Congress association

Bon Maharaj Engineering College, Vrindavan

Mathura Uttar Prades

Dec. 8-9, 2012

5

Chemselective recations of 2-methylbenzo[h]naphthyridines

 

International conference on herbal & synthetic drug studies

Abeda Inamdar Sr. College, Pune

12-02-2014

6

Chemselective recations of 2-methylbenzo[h]naphthyridines

 

International conference on herbal & synthetic drug studies ;

Abeda Inamdar Sr. College, Pune

12-02-2014

7

New methods  for solution phase parallel synthesis

 

Global opportunities for latest developments in chemistry and Technology,

Dept of Chem

North Maharashtra Uni. Jalgaon

6-8 Feb. 2014

8

Reactions of a-acetyl-g-butyro lactone with 2-aminoheterocylics

 

European Colloquium on Heterocyclic Chemistry

Bari, Italy

Sept.2-6, 2006

9

Synthesis of novel pyridine derivatives , 26-28th Nov. 1998

XVIIth Conference of Indian of Indian Council of Chemists, Chennai

Uni of Madras

Chennai

26-28th Nov. 1998

 

 Papers In National Conferenc :

1

The strength love is trust

 

National Conference

2

M.J. College, Jalgaon

29-30th Oct. 2004

2

Synthesis of Aroylacetonitrile using mortor & pest January,

90th Indian Science Congress Conference,

Bangalore, India

Jan. 3-7,th 2003

3

Novel route for synthesis of 4-aroyl & 4-aminopyrimidines.

91st Indian Science Congress Conference,

Chandigarh, India, Panjab

Jan. 3-7th ,2004

4

Synthesis of new fused pyrimidines

92nd Indian Science Congress conference ISCA 2005

Nirma University

Ahmedabad

Jan.3-7th, 2005

5

Synthesis of Anti-oxidant activity of new theino-heterocyclic compounds 

94th Indian Science Congress

 

Andra University Vishkhapatanm

Jan 3-7th , 2008

6

Effect of substituent on absorption & fluoresce properties of pyrazolo[3,4-b] pyralo[2,3-d]pyridines

96th Indian Science Congress

 

North Hill Eastern Uni. Shillong, Assam, India ,

Jan. 3-7th 2009

7

Synthesis and study of biological activities of new indanaone derivatives

96th Indian Science Congress

 

Trivendrum,

Kerala, January,

Jan. 3-7, 2010

8

Sulfamic acid mediated  one-pot synthesis of amide acid derivatives

 

99th Indian Science Congress

 

KITT University

Bhubaneswar, Orissa

Jan 3-7, 2012

9

 Applications of Chemistry

 

UGC &  SHGM College,

Kopergaon, Dist-Ahamednagar

UGC & SHGM College, Kopergaon

Feb. 11-13, 2012

10

Sulfamic acid mediated efficient one-pot synthesis of novel  5-substituted 1,3,4-thiadiazol-2-ylcarbamoyl) aliphatic amide acid derivatives

Perspective of Organic Synthesis

 

Dept of Chemistry

Uni of

Pune-07

March 24, 2012

11

An efficient micro wave -assisted Suzuki cross-coupling react ions on quinoline derivatives in water and study the electronic effects

Indian Science Congress association ISCA 2013

 

Calcutta University, Kolkata

 

Jan. 3-7, 2013

12

An efficient micro wave -assisted Suzuki cross-coupling react ions on quinoline derivatives in water and study the electronic effects

Indian Science Congress association ISCA 2013

Calcutta University, Kolkata

 

Jan. 3-7, 2013

13

Synthesis & Insecticidal activity of novel triazene & triaza indacene pyrazole derivatives 

Recent Advances on Chemical Sciences & technology

 

NMU, Jalgaon

Sept 21, 2013

14

Synthesis & Insecticidal activity of novel triazene & triaza indacene pyrazole derivatives 

Recent Advances on Chemical Sciences & technology

NMU, Jalgaon

Sept 21, 2013

15

Synthesis and Fluorescence Properties of Donor-Acceptor Substituted Novel Thieno[3, 2-c]pyridine;

National symposium on functional applications of colorants ;

ICT, Mumbai

29-30 Oct 2013

16

Synthesis and Fluorescence Properties of Donor-Acceptor Substituted Novel Thieno[3, 2-c]pyridine;

National symposium on functional applications of colorants ;

ICT, Mumbai

Oct 29-30 2013

17

Synthesis of insecticidal activity of novel triazene & triaza-s-indacene pyrazole derivatives;

National conference on Redefine  role of chemistry in modern science

VN Naik College, Nashik

Feb, 13-14, 2014

18

Synthesis of ?-formyl-?-butyrolactone and a-fornyl-?-valerolactone

 

National symposium on functional applications of colorants

ICT, Mumbai

OCT 16-17,2014

19

Synthesis of Novel thiazole substituted cytosine & Uracil analogues

 

National Seminar on Chemistry for overall development

KSKW College, CIDCO, Nashik

Jan 16-17,  2015

20

Synthesis of benzothienopyridine & benzothienopyrimidine derivatives as good antioxidents;

National seminar on Recent trends of research in chemistry

ASC College Rahata

A`Nagar

Feb 13-14,  2015

21

Synthesis of thieno[3, 2-c] pyridine study of their photophyscial properties with respective to donor-acceptor substitut`s

Indian Science Congress, Mysure, Karnatak ;

 

Mysure University

Karnatak

Jan. 3-7 2016

22

Effect of substituent at imino gr. on phophysical properties of pyrazolone azomethine derivatives

 

Institute of Chemical technology

Matunga Mumbai

 

National

 

Oct. 11-12, 2012

23

New route for the synthesis of 4-aminopyrazoles

87th Indian Science Congress conference,

Uni  Pune

3-7, January 2000

24

Synthesis of New cytosine  derivatives

National Symposium on New Trends in Synthetic Organic Chemistry

KTHM College, Nashik-02

 

 

 Conference/ Workshop Attended :

1

 Fused heterocyles with 3-(2S) and 3-(2R) side chain: synthesis and Biological activity evaluation ;Nov.

Innovation in Chemistry

BCUD, Uni. Pune

KTHM College, Nashik

10-11, 2008

2

Synthesis of New Antimalarial drugs such as 2-methy lbenzo[h][1,6 ]naphtahridines

BCUD, UoP

Ahmednagar College

16/4/2013

3

Synthesis of New Antimalarial drugs such as 2-methy lbenzo[h][1,6 ]naphtahridines

BCUD, UoP

Ahmednagar College

16/4/2013

4

Innovation in chemistry

BCUD UoP ,

 

KTHM , Nashik,

Nov. 24-25, 2009

5

Innovation in chemistry

 

BCUD UoP & KTHM College

Uni. Pune, & KTHM , Nashik,

Nov. 24-25,2010

6

Synthesis of Biologically active  Quinolines   

Innovation 2007 ;

 

Uni Pune

19/11/2007

7

Resolution of aminoethyl-4-hydroxy methylquinolone using disterimeric salt formation

INNOVATION 2014

University of Pune

 

Dept of Chem

Uni Pune

2-04-2014

8

Synthesis using grind stone technology

Green Chemistry,

KANMS ASC College, satana

UGC & Satana College

 

15-16 Jan. 2010

9

Green reactions & atom economy;

VN Naik College,

 Nashik-02

 

BCUD, UoP &

VN Naik College

21/01/2011

10

Sensitizing students to green chemistry;

 

Environmental Conservation & sustainable Development

RNC Bytco College, Nashik Road Nashik

Dec. 28-29, 2012

11

Applications of Green Chemistry Sensitizing Students for Green Chemistry;

Importance of green Chemistry

RNC Arts, Bytco College, N.Road

26-09-2014

12

Synthesis of new tetracyclic indeno thienopyrimidine derivatives

State level seminar on New trends in modern Chemistry

 

ASC College Kalwan

18-19-Dec.014

13

Applications of Green Chemistry Sensitizing Students for Green Chemistry

Importance of green Chemistry

RNC Arts, Bytco College, N.Road

26-09-2014

14

Reaction of Sodim  salt of g-butyrolactone  with 2-aminoheterocylic compounds

Recent trends in Chemical research

 

VN Naik College, Nashik

13-2-13 Jan.2015

15

Reactions of a-acetyl-g-butyrolactone with 2-aminopridines

National conference on Emerging trends in Chemical science

 

Adv.M.N. Deshmukh A.S.C. College, Rajur, Tal-Akole, A`nagar

30-31 Jan. 2015

16

Human touch of Chemistry

 

State level Seminar on Recent Development & Future Challenges in Chemical Sciences

ASC College Nadgaon

 

22-23 Jan. 2016

17

Chemistry around us

 

International Conference

Bytco College

Nashik Road

2017

18

Use of IR spectroscopy: New Dimensions, Chair the session & Deliver lecture 

 

Spectroscopic Trends in Organic & Inorganic Chemistry,

SSGM College, Kopargoan

24-25 Feb. 2009

19

Applications of IR

 

Organic spectroscopy

KKW A.S.C. College, Pimpalgaon (B), Dist-Nashik

17-01-2011

20

Atom Economy

 

State level conference on Green Chemistry

Adv. M.N. Deshmukh ASC College, Akole Dist-A`Nagar

10-01-2011

21

New Advances in UV spectroscopy Chair person

 

Spectroscopic Techniques

& Applications

 

A.S.C. College Lasalgaon

10-02-2012

22

Advances in synthetic & Applied Chemistry 

 

Advances in synthetic

 and applied Chemistry

 

UGC & Sangmner

College

Sept 6-8, 2012

23

Applications of spectroscopy in Chemistry

NMR spectroscopy

Radhabai Kale Mahila

Mahavidyalaya,

A`Nagar

Feb 2014

24

New synthetic methods in organic chemistry

 

State level seminar on Applications of synthetic chemistry,

MVP Samaj

ASC College

Dindori

1-2 March 2013

 

 Ph.D. Guidance :

v No. of students completed Ph.D.: 11

 

Sr. No.

Name of Student

Research Topic

Degree Awarded

1

Mr. Bhausaheb Ghotekar  K.

Synthesis of Novel Heterocyclic such as Quinolines and Pyrimidines

Feb 2009

2

Mr. Kazi Muddassar  A.

Synthesis of Thieno pyridines/ pyrimidines and Evaluation of their Anti-Oxidant activities.

May 2009

3

Patil Shivaraj P.

Synthesis of fused pyridines having Intractable side chain and study of their biological activity.

Oct 2009

4.

Dr. Pagar Balasaheb

Synthesis of novel Benzo[h][1,6]naphthyridine and Cyclopenta[a]phenanthren-7-ylsulfanyl derivatives: Study of their biological activities and photophysical properties

Feb 2011

5

Dr.Dinesh Bhavsar

Facile synthesis of pyrazolo annulated heterocyles and attachment of linkers to new pyazolopyridine and pyridines

Oct 2012

6

Dr. Ravi Janrao

Suzuki-Miyora Cross coupling reactions on heterocyclic nucleus in presence of unmasked functional group: synthesis of benzo[h][1,6] naphthyridines

Dec 2012

7

Dr. Prashant Nikam

 

Synthesis of New Nicotinonitrile derivatives and Indeno-pyrazolo[3,4-b] pyridine and Evaluation of their photophysical and biological activities

30-01-2014

8

Dr. Shrikant Kanwade

Synthetic  applications of o-aminothiophene dicarbonitrile and o-aminothiophene dicarbox amide precursors: Synthesis of new thienopyridine, thienopyrimidine derivatives and study of their biological activities

13-08-2014

9

Dr. Sachin Gangurde

 

Synthesis of azo derivatives from pyrazolone, 2-aminothiophene and 4-hydroxyquinolone: Study of their photophysical properties and applications in colour chemistry

 

14-11-2014

10

Dr. Gorakh Shinde

 

Synthesis and Biological evaluation of few optically pure compounds containing Quinolinones, Pyrazolothio- phenols and Napthylethylamine frameworks.

12/01/2013

11

Dr. Sunil Chavan

Synthesis of new derivatives of thiophene and thiophene fused heterocycles and evaluation of their photophysical and biological activities.

May 2016

 

·         No.of  Students presntly working for Ph.D. : 06

 

Sr.

No.

Name of Student

Date of Registration

Research Topic

1

Chavan S.M

2013

Synthesis of Pyrazole and thiophene derivatives and study of their biological activity

2

Madhukar Shinde

2014

Synthesis of transition metal complexes of Schiff’s  bases and to Study their biological

Activities

3

Kunal Dingore

2014

Synthesis and study of photo physical properties of linear heterocyclic molecules

4

Rahul Watpade

2015

Synthesis of  Benzo[h][1,6]naphthyridine derivatives and study of their anti-malarial activities

5

Kunal Jagatap

2015

Synthesis, Characterization of Novel Pyrimidine Derivatives & Evaluation of their Biological Activities and Process Development of few Endothelin Receptor Antagonist Drugs

6

Sanjay Deshmuk

2015

Synthesis of Thiazole containing Novel Heterocyclic compound and their Biological evaluation

·        No. of students awarded M.Phil.

 

Sr. No.

Name of Student

 Research Topic

Degree Awarded/working  

1

Smt. J. D. Varade

Eco Friendly Organic Synthesis: Use of Solvent Free Neat and Microwave Techniques for Cytosines, Uracils Synthesis

2009

2

Smt. Pushpa

Patil

Green synthesis of Thieno-Pyridine, Thieno-Pyrimidines and Evaluation of their Anti-oxidant Activity

2008

3

Mr Pankaj Aware

Synthesis of new pyrido[1,2-a]pyrimidine, pyrimidine and 5-cyano uracil  derivatives

 

 2016

4

Mr. Madan patil

Synthesis and characterization of Oxazole, Thiazole and pyrazolopyridine Derivatives

2016

5

Poonam patil

Synthetic utility of Gewald reaction: Synthesis of thiozaoles 

Thesis submitted

6

Mrs. S.M. Tambade

Development of Reagents for conversion of aldehyde to alcohols

 

Working

 

 Major/ Minor Research Project :

Research Projects: Completed/ Ongoing/ submitted

·         Project Completed: CSIR- 01; UGC Major =02; UGC Minor =3; BCUD=03

Sr. No.

Title of the research Project

Duration & Amount

Major

/Minor

Funding Agency

1

Synthesis of New Benzo[h] naphthyridines and to study the Influence of substitutes on Anti- Malarial Activity

2009-13

13, 26, 000/-

Major

 

CSIR

New Delhi

2

Synthesis of Novel Indenothiophenes and Study their Antioxidant activities

2012-13

2,80,000/-

Minor

 

BCUD, Uni. Pune, Pune

 

3

Synthesis of Benzo [h] naphthyridines having 3-Substituded Ethyl Side Chain and Study of Their Anti-Malarial Activities.

2009-12

6, 89, 000/-

Major

 

UGC

New Delhi

 

4

Synthesis and Evaluation of Anti-malarial, CNS and   Antifungal Activity of Novel Heterocyclic Compounds Such As Quinolines and  Pyrimidines

 

January 2005-

December 2007

5,81,100/-

 

Major

 

UGC, Major

New Delhi

5

Fused heterocyles with active substituent:  Synthesis and Biological  activity evaluation

 

Jan. 2007

Rs.2,00,000/-

 

Minor

BCUD,

Uni. of Pune

6

Synthesis of Biologically active Quinolines

 

1998-2000

Rs. 40000/-

 

Minor

UGC, WRO, Pune

7

Synthesis of clinically useful fused pyrimidine derivatives

Feb. 2002-04

Rs.40,000/-

Minor

UGC, WRO, Pune

·        Ongoing projects

 

1

Synthesis of polysubstituted thiophene and thiazole derivatives and study of their biological activities

2016-18

Rs. 2,50,000/-

BCUD, SPPU, Pune

BCUD, SPPU, Pune

Sponsored Research by  Megafine Pharmacaeutical PVT LTD, Dindori, Nashik

Dr. Gorakh Shinde

 

Synthesis and Biological evaluation of few optically pure compounds containing Quinolinones, Pyrazolothio- phenols and Napthylethylamine frameworks.

12/01/2013

 

Kunal Dingore

Synthesis and study of photo physical properties of linear heterocyclic molecules

2014

 

 

 Course Conducted :

UGC Sponsored Community College in Community College in Analytical Techniques for Pharmaceuticals (Skill Sector Life Science)

UGC Sponsored  Carrier Oriented Course in Instrumental Techniques in Analytical Chemistry (Skill Sector Life Science)

 

 Other :

Ø Fellowship/ Award

 

1.

OeAD,  Scholarship for Guest Scientist in Austria, Europe ,  1996-97

2.

UGC Teacher Fellowship Under , Faculty Improvement  Program (FIP); 1999-2001

3.

Best Teacher Award of University of Pune, Pune-411007, February  2009

4.

Best Teacher Award by (SAVANA Nashik) Sarvgenic Vachnalay, Nashik; Sept. 2010

5.

Best Chemistry Teacher Award by Tata Chemicals 2011

(Award partners: Tata group, Indian of Chemistry Teacher Association Human Touch of Chemistry,  IIT, CSIR, IIT, NCL), Jan. 2011

6.

Prof. N. S. Narasimhan endowment Award, 2012 for Research at College level by Prof. Narashimhan Trust, Dept of Chemistry, University of Pune; Feb 2012

7.

Shikshak Ratna Purshkar by Maharshtra Rajya Patrakar Sangh, Sept. 2012

Ø Co-ordinator of  the  Funding Schemes of UGC & DST  New Delhi                          

  • College with Potential  for Excellence (CPE, 3rd  Phase)
  • Dept. of Science & technology (DST)
  • Bachelor of Vocational (B.Voc.)
  • Community College
  • Carrier oriented Courses

 

Ø  Extra -Curricular  Activities:

 

·         Board of study member of Chemistry (BOS),  University of Pune, 2011-2015

·         Member of Chemistry syllabus  revision committee for S.Y. /T.Y. /M. Sc. (2013-15).

·         Secretary of Cluster 3 (Students centric) programme of Pune University for Nashik zone.

·         Chairman, M.Sc. Organic Chemistry, University of Pune (2009-2011, 2015-17)

·         Co-ordinator of S.Y.B.Sc University Exam. University of Pune, (2005-2008)

·         Co-ordinator of Minority coaching classes for competitive examinations  sponsored

by UGC, New Delhi (2002)

·         Chairman and member of Local Inquiry Committees of University

·         Co-ordinator of Cyber Security, Human Rights and Skill Development

Courses for all PG classes.

·         300 Projects Human values and Rights were done by  PG students

·         Co-ordinator of NAAC criterion 3

 

Ø Events organized (Co-ordinator) in College:

  1. State level workshop “on Over view of analytical Instruments Sponsored by BSR Technologies, MICD, Ambad (13 August 2016)

2.      Faculty Development programme for Senior Chemistry  Teachers UGC-Academic  staff college, UoP (August 5-10, 2013)         

3.      Workshop on credit system syllabus framing workshop (July 6, 2013).

  1. One day National Conference on ‘Advances and Opportunities in Chemical Sciences’ on Saturday  in collaboration with Royal Society of Chemistry
  2. Workshop on “Hands on training on sophisticated instrument” sponsored by Shumadzu Analyticals, 23-26, March 2015.

6.      Advanced Spectroscopic techniques, funded by Indian Academy of  Sciences, Bangalore, Indian National Science Academy, New Delhi, The National Academy of Sciences, India, Allahabad 3-5th  Feb 2013

7.      National level workshop on Analytical Instruments, Funded by  Shimadzu Analytical (India) Pvt. Ltd., Mumbai 23-25 Aug.2012,

8.      Advances and Opportunities in Chemical Sciences, funded by Royal Chemical Society (West India Section); 20-10-2012

9.      National level conference on Interface between Academia and Industries, 26-28 Dec. 2007, UGC, New Delhi

10.  State level seminar on Interface between Academia and Industries, Jan.2004, Indian Chemistry Teacher association CT, Mumbai,

11.  State  level conference on Computer applications in chemistry

                   Nov. 2001, University of Pune

12.  Workshop on State (SLET) Eligibility Exam Centre, Uni. of Pune-07 Nov. 2007 Dec 2002   & Dec. 2004.

13.  Zonal Level Research Project Competition, Avishkar, December 8, 2011, December 1, 2012, December 7, 2013

14.  Avishkar Orientation Workshops: Dec.  9, 2011; Dec. 21, 2012;  Dec.  24, 2013;

                                                                               Sept. 3, 2015, Oct 5, 2015; Dec. 22, 2016

15.  Innovations : November 21-22,  2010 &  September 30, 2016

Ø Industrial Training organized: 

·         Training to Community College students on handling of instrument in BSR Technology, MIDC Ambad May 2016.

·         Training to M.Sc. students in VSL, MIDC, Gonde, Igatpuri, Nashik

Ø Industrial/ Institutional  visits organized:

1.      Regional Forensic Lab Nashik-03, Forensic Awareness Week Jan  30-Feb. 2012

2.      Visit to Niphad Sahakari Sakhar Karkhana  2002, 2003, 2004

3.      National Chemical Laboratory & Dept of Chemistry, University of Pune, 2005

4.      Indian Institute of Science & Research (IISER) Pune, 2013

5.      Indian Institute of Technology (IIT), Powai (Mumbai) 2011

6.      Mega fine pharmaceuticals PVT LTD, Lakhamapur, Dindori

7.      Vadivara Specialty Chemicals, PVT LTD, MIDC Gonde, Igatpuri  2014, 2015, 2016

8.      Glenmark, Sinnar, 2016

9.      Global Chem, MIDC, Sinnar, 2016

 

Ø Establish Academic & Research Linkages and  Collaborations

 

·         Dept. of Organic and Bio-organic Chemistry, University of Graz, Austria,

  • Microcare Laboratory and TRC, Unapani Road, Lal Darwaja, Surat (Gujarat), India
  • Megafine Pharmacuticals Pvt Ltd, Lakhmapur, Dindori, Nashik
  • Shimadzu analyticals Pvt.LTd, Mumbai
  • BSR Technologies, MIDC Ambad, Nashik
  • Dept of Chemistry, University of Pune, Pune-411007
  • Department of Zoology, and Bio-technology KHM College, Nashik-02
  • Baha`i Academy, Pachgani (Mahabaleswar)
Back
 

Designed and Developed by - Computer Science Department